19002083. POSITIVE MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 (Vanderbilt University)
POSITIVE MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4
Organization Name
Inventor(s)
Craig W. Lindsley of Brentwood TN US
Darren W. Engers of Brentwood TN US
Kayla J. Temple of Spring Hill TN US
Alison R. Gregro of Mount Juliet TN US
Alexa E. Richardson of Nashville TN US
Madeline F. Long of Nashville TN US
POSITIVE MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4
This abstract first appeared for US patent application 19002083 titled 'POSITIVE MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4
Original Abstract Submitted
Deuterium-labeled 4-((2,3-dihydrobenzo[b][1,4]dioxin-6-yl)oxy)piperidines substituted with pyrrolo[3,4-b]pyridin-5-one, furo[3,4-b]pyridin-5(7H)-one, or [1,2,4]triazolo[4,3-a]pyrimidin-3(2H)-one are positive allosteric modulators of the muscarinic acetylcholine receptor M(mAChR M) and may have use in treating neurological and psychiatric disorders associated with muscarinic acetylcholine receptor dysfunction.